6HXR
Human PARP16 (ARTD15) IN COMPLEX WITH EB-47
Summary for 6HXR
Entry DOI | 10.2210/pdb6hxr/pdb |
Descriptor | Mono [ADP-ribose] polymerase PARP16, 2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide (2 entities in total) |
Functional Keywords | transferase, adp-ribose, parp16, artd15, adp-ribosylation, eb-47, inhibitor complex |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 3 |
Total formula weight | 101821.78 |
Authors | Karlberg, T.,Pinto, A.F.,Thorsell, A.G.,Schuler, H. (deposition date: 2018-10-18, release date: 2019-10-30, Last modification date: 2024-01-31) |
Primary citation | Karlberg, T.,Pinto, A.F.,Thorsell, A.G.,Schuler, H. Human PARP16 (ARTD15) IN COMPLEX WITH EB-47 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.9 Å) |
Structure validation
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