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6HWS

Keap1 - inhibitor complex

Summary for 6HWS
Entry DOI10.2210/pdb6hws/pdb
DescriptorKelch-like ECH-associated protein 1, 1,2-ETHANEDIOL, 2-[[4-[2-hydroxy-2-oxoethyl-(4-methoxyphenyl)sulfonyl-amino]-3-phenylmethoxy-phenyl]-(4-methoxyphenyl)sulfonyl-amino]ethanoic acid, ... (5 entities in total)
Functional Keywordskeap1, kelch-domain, nrf2, neurodegenerative, inhibitor, peptide binding protein
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight32548.08
Authors
Talapatra, S.K.,Kozielski, F.,Wells, G.,Georgakopoulos, N.D. (deposition date: 2018-10-13, release date: 2019-10-30, Last modification date: 2024-01-24)
Primary citationTalapatra, S.K.,Kozielski, F.,Wells, G.,Georgakopoulos, N.D.
Keap1-inhibitor complex
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

222036

PDB entries from 2024-07-03

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