6GTU
17beta-hydroxysteroid dehydrogenase 14 variant T205 in complex with fragment J6
Summary for 6GTU
Entry DOI | 10.2210/pdb6gtu/pdb |
Related | 6EMM 6GTB |
Descriptor | 17-beta-hydroxysteroid dehydrogenase 14, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, N-(1,3-benzodioxol-5-ylmethyl)cyclopentanamine, ... (6 entities in total) |
Functional Keywords | fragments, soaking, 17b-hsd14, oxidoreductase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 29751.07 |
Authors | Bertoletti, N.,Heine, A.,Marchais-Oberwinkler, S.,Klebe, G. (deposition date: 2018-06-19, release date: 2019-07-03, Last modification date: 2024-01-17) |
Primary citation | Bertoletti, N.,Braun, F.,Zara, L.,Metz, A.,Heine, A.,Marchais-Oberwinkler, S.,Klebe, G. X-ray Crystallographic Fragment screening and Hit Optimization To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.25 Å) |
Structure validation
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