6G88
Crystal structure of Enterococcus Faecium D63r Penicillin-Binding protein 5 (PBP5fm)
Summary for 6G88
Entry DOI | 10.2210/pdb6g88/pdb |
Related | 6G0K |
Descriptor | Low affinity penicillin-binding protein 5 (PBP5), (2R)-2-[(1R)-1-{[(2Z)-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(hydroxyimino)acetyl]amino}-2-oxoethyl]-5-({2-oxo-1-[(3R)-pyrrolidin-3-yl]-2,5-dihydro-1H-pyrrol-3-yl}methyl)-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, SULFATE ION (3 entities in total) |
Functional Keywords | penicillin-binding, ceftobiprole, enterococcus faecium, antibiotic resistance, antibiotic |
Biological source | Enterococcus faecium (Streptococcus faecium) |
Total number of polymer chains | 3 |
Total formula weight | 214129.26 |
Authors | Sauvage, E.,El Gachi, M.,Herman, R.,Kerff, F.,Charlier, P. (deposition date: 2018-04-08, release date: 2019-04-24) |
Primary citation | Sauvage, E.,El Gachi, M.,Kerff, F.,Herman, R.,Verlaine, O.,Amoroso, A.,Page, M.G.P.,Joris, B.,Charlier, P. Structural basis of inactivation of Enterococcus faecium penicillin binding protein 5 by ceftobiprole. To Be Published, |
Experimental method | X-RAY DIFFRACTION (3.3 Å) |
Structure validation
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