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6G3V

Crystal structure of human carbonic anhydrase I in complex with the inhibitor famotidine

Summary for 6G3V
Entry DOI10.2210/pdb6g3v/pdb
DescriptorCarbonic anhydrase 1, ZINC ION, famotidine, ... (5 entities in total)
Functional Keywordslyase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight58898.39
Authors
Ferraroni, M.,Supuran, C.T.,Angeli, A. (deposition date: 2018-03-26, release date: 2018-11-28, Last modification date: 2024-01-17)
Primary citationAngeli, A.,Ferraroni, M.,Supuran, C.T.
Famotidine, an Antiulcer Agent, Strongly InhibitsHelicobacter pyloriand Human Carbonic Anhydrases.
ACS Med Chem Lett, 9:1035-1038, 2018
Cited by
PubMed: 30344913
DOI: 10.1021/acsmedchemlett.8b00334
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.69 Å)
Structure validation

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