6G3Q
Crystal structure of human carbonic anhydrase II in complex with the inhibitor famotidine
Summary for 6G3Q
Entry DOI | 10.2210/pdb6g3q/pdb |
Descriptor | Carbonic anhydrase 2, ZINC ION, famotidine, ... (5 entities in total) |
Functional Keywords | lyase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 29786.03 |
Authors | Ferraroni, M.,Supuran, C.T.,Angeli, A. (deposition date: 2018-03-26, release date: 2018-11-28, Last modification date: 2024-01-17) |
Primary citation | Angeli, A.,Ferraroni, M.,Supuran, C.T. Famotidine, an Antiulcer Agent, Strongly InhibitsHelicobacter pyloriand Human Carbonic Anhydrases. ACS Med Chem Lett, 9:1035-1038, 2018 Cited by PubMed: 30344913DOI: 10.1021/acsmedchemlett.8b00334 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.01 Å) |
Structure validation
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