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6FZJ

PPAR gamma mutant complex

Summary for 6FZJ
Entry DOI10.2210/pdb6fzj/pdb
DescriptorPeroxisome proliferator-activated receptor gamma, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, (2~{S})-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]-2-[[2-(phenylcarbonyl)phenyl]amino]propanoic acid, ... (6 entities in total)
Functional Keywordsnuclear receptor, transcription
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains4
Total formula weight67297.43
Authors
Rochel, N. (deposition date: 2018-03-14, release date: 2019-02-13, Last modification date: 2024-01-17)
Primary citationRochel, N.,Krucker, C.,Coutos-Thevenot, L.,Osz, J.,Zhang, R.,Guyon, E.,Zita, W.,Vanthong, S.,Hernandez, O.A.,Bourguet, M.,Badawy, K.A.,Dufour, F.,Peluso-Iltis, C.,Heckler-Beji, S.,Dejaegere, A.,Kamoun, A.,de Reynies, A.,Neuzillet, Y.,Rebouissou, S.,Beraud, C.,Lang, H.,Massfelder, T.,Allory, Y.,Cianferani, S.,Stote, R.H.,Radvanyi, F.,Bernard-Pierrot, I.
Recurrent activating mutations of PPAR gamma associated with luminal bladder tumors.
Nat Commun, 10:253-253, 2019
Cited by
PubMed: 30651555
DOI: 10.1038/s41467-018-08157-y
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.011 Å)
Structure validation

217705

数据于2024-03-27公开中

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