6FUK
Crystal structure of UTX complexed with 5-carboxy-8-hydroxyquinoline
Summary for 6FUK
Entry DOI | 10.2210/pdb6fuk/pdb |
Descriptor | Lysine-specific demethylase 6A, MANGANESE (II) ION, 8-hydroxyquinoline-5-carboxylic acid, ... (8 entities in total) |
Functional Keywords | jumonji demethylase, inhibitor, oxidoreductase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 61098.40 |
Authors | Esposito, C.,Sledz, P.,Caflisch, A. (deposition date: 2018-02-27, release date: 2018-10-10, Last modification date: 2024-01-17) |
Primary citation | Esposito, C.,Wiedmer, L.,Caflisch, A. In Silico Identification of JMJD3 Demethylase Inhibitors. J Chem Inf Model, 58:2151-2163, 2018 Cited by PubMed: 30226987DOI: 10.1021/acs.jcim.8b00539 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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