6FRX
PKA variant as Aurora B mimic in complex with a dianilinopyrimidine inhibitor
Summary for 6FRX
Entry DOI | 10.2210/pdb6frx/pdb |
Descriptor | cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha, ~{N}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamide, ... (4 entities in total) |
Functional Keywords | protein kinase, surrogate model, catalytic domain, transferase |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 43448.69 |
Authors | |
Primary citation | Engh, R.A.,Kazi, A.A. PKA variant as Aurora B mimic in complex with a dianilinopyrimidine inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.88 Å) |
Structure validation
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