6FQT

Crystal structure of CREBBP bromodomain complexd with DR46

Summary for 6FQT

• Entry DOI: 10.2210/pdb6fqt/pdb
• Descriptor: CREB-binding protein, ~{N}-[3-(5-ethanoyl-2-ethoxy-phenyl)-5-(1-methylpyrazol-3-yl)phenyl]furan-2-carboxamide (3 entities in total)
• Functional Keywords: inhibitor, bromodomain, transferase
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15082.28

Authors

Zhu, J.,Caflisch, A. (deposition date: 2018-02-14, release date: 2019-03-13, Last modification date: 2024-01-17)

• Primary citation: Zhu, J.,Caflisch, A.; Crystal structure of CREBBP bromodomain complexd with DR46; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.8 Å)