6FGD
Crystal structure of Gephyrin E domain in complex with Artemether
Summary for 6FGD
Entry DOI | 10.2210/pdb6fgd/pdb |
Descriptor | Gephyrin, CALCIUM ION, PHOSPHATE ION, ... (9 entities in total) |
Functional Keywords | antimalarial compound, scaffolding protein, moonlighting protein, inhibitory neurotransmission, structural protein |
Biological source | Rattus norvegicus (Rat) |
Total number of polymer chains | 1 |
Total formula weight | 48111.32 |
Authors | Kasaragod, V.B.,Schindelin, H. (deposition date: 2018-01-10, release date: 2019-01-16, Last modification date: 2024-01-17) |
Primary citation | Kasaragod, V.B.,Hausrat, T.J.,Schaefer, N.,Kuhn, M.,Christensen, N.R.,Tessmer, I.,Maric, H.M.,Madsen, K.L.,Sotriffer, C.,Villmann, C.,Kneussel, M.,Schindelin, H. Elucidating the Molecular Basis for Inhibitory Neurotransmission Regulation by Artemisinins. Neuron, 101:673-689.e11, 2019 Cited by PubMed: 30704910DOI: 10.1016/j.neuron.2019.01.001 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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