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6FDZ

Unc-51-Like Kinase 3 (ULK3) In Complex With Momelotinib

Summary for 6FDZ
Entry DOI10.2210/pdb6fdz/pdb
DescriptorSerine/threonine-protein kinase ULK3, Momelotinib (3 entities in total)
Functional Keywordskinase inhibitor dfg-out, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight32354.44
Authors
Mathea, S.,Salah, E.,Moroglu, M.,Scorah, A.,Pike, A.C.W.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Huber, K.,Knapp, S. (deposition date: 2017-12-27, release date: 2018-08-01, Last modification date: 2024-01-17)
Primary citationMathea, S.,Salah, E.,Moroglu, M.,Scorah, A.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Huber, K.,Knapp, S.
Unc-51-Like Kinase 3 (ULK3) In Complex With Momelotinib
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.55 Å)
Structure validation

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