6FDC
Crystal structure of the PDE4D catalytic domain in complex with GEBR-32a
Summary for 6FDC
Entry DOI | 10.2210/pdb6fdc/pdb |
Descriptor | cAMP-specific 3',5'-cyclic phosphodiesterase 4D, ZINC ION, MAGNESIUM ION, ... (7 entities in total) |
Functional Keywords | pde4, catalytic domain, inhibitor, gebr, hydrolase |
Biological source | Homo sapiens (Human) |
Cellular location | Apical cell membrane : Q08499 |
Total number of polymer chains | 2 |
Total formula weight | 80501.33 |
Authors | Prosdocimi, T.,Donini, S.,Parisini, E. (deposition date: 2017-12-22, release date: 2018-05-16, Last modification date: 2024-05-08) |
Primary citation | Prosdocimi, T.,Mollica, L.,Donini, S.,Semrau, M.S.,Lucarelli, A.P.,Aiolfi, E.,Cavalli, A.,Storici, P.,Alfei, S.,Brullo, C.,Bruno, O.,Parisini, E. Molecular Bases of PDE4D Inhibition by Memory-Enhancing GEBR Library Compounds. Biochemistry, 57:2876-2888, 2018 Cited by PubMed: 29652483DOI: 10.1021/acs.biochem.8b00288 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.45 Å) |
Structure validation
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