6E7R
Heterodimer of the GluN1b-GluN2B NMDA receptor amino-terminal domains bound to allosteric inhibitor 93-4
Summary for 6E7R
Entry DOI | 10.2210/pdb6e7r/pdb |
Descriptor | Glutamate receptor ionotropic, NMDA 1, Glutamate receptor ionotropic, NMDA 2B, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total) |
Functional Keywords | nmda receptor, ion channel, allosteric modulation, extracellular domain, transport protein |
Biological source | Xenopus laevis (African clawed frog) More |
Total number of polymer chains | 4 |
Total formula weight | 172886.77 |
Authors | Regan, M.C.,Furukawa, H. (deposition date: 2018-07-27, release date: 2019-01-30, Last modification date: 2023-10-11) |
Primary citation | Regan, M.C.,Zhu, Z.,Yuan, H.,Myers, S.J.,Menaldino, D.S.,Tahirovic, Y.A.,Liotta, D.C.,Traynelis, S.F.,Furukawa, H. Structural elements of a pH-sensitive inhibitor binding site in NMDA receptors Nat Commun, 10:321-, 2019 |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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