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6DN5

SPRY domain-containing SOCS box protein 2 complexed with WDINNN(BAL) cyclic peptide inhibitor

Summary for 6DN5
Entry DOI10.2210/pdb6dn5/pdb
Related PRD IDPRD_002313
DescriptorSPRY domain-containing SOCS box protein 2, WDINNN(BAL) cyclic peptide inhibitor, SULFATE ION, ... (4 entities in total)
Functional Keywordsproteasomal degradation, nitric oxide, inhibitor, immune system, immune system-inhibitor complex, immune system/inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight24887.61
Authors
Law, R.H.P.,Caradoc-Davies, T.T.,Norton, R.S. (deposition date: 2018-06-06, release date: 2019-04-17, Last modification date: 2020-01-08)
Primary citationSadek, M.M.,Barlow, N.,Leung, E.W.W.,Williams-Noonan, B.J.,Yap, B.K.,Shariff, F.M.,Caradoc-Davies, T.T.,Nicholson, S.E.,Chalmers, D.K.,Thompson, P.E.,Law, R.H.P.,Norton, R.S.
A Cyclic Peptide Inhibitor of the iNOS-SPSB Protein-Protein Interaction as a Potential Anti-Infective Agent.
ACS Chem. Biol., 13:2930-2938, 2018
Cited by
PubMed: 30226743
DOI: 10.1021/acschembio.8b00561
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

数据于2024-03-27公开中

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