6DB0
N-Terminal bromodomain of Human BRD2 with a Tetrahydroquinoline analogue
Summary for 6DB0
Entry DOI | 10.2210/pdb6db0/pdb |
Descriptor | Bromodomain-containing protein 2, SULFATE ION, 1-[(2S,4R)-4-[(2-chlorophenyl)amino]-2-methyl-6-(1H-pyrazol-3-yl)-3,4-dihydroquinolin-1(2H)-yl]ethan-1-one, ... (6 entities in total) |
Functional Keywords | bet, brd2, bromodomain, inhibitor, complex, transcription, transcription-inhibitor complex, transcription/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 3 |
Total formula weight | 49610.67 |
Authors | White, S.W.,Yun, M. (deposition date: 2018-05-02, release date: 2019-11-13, Last modification date: 2023-10-04) |
Primary citation | White, S.W.,Yun, M. N-Terminal bromodomain of Human BRD2 with a Tetrahydroquinoline analogue To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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