6CCF

Crystal Structure of the Human CAMKK1A in complex with Hesperadin

Summary for 6CCF

• Entry DOI: 10.2210/pdb6ccf/pdb
• Descriptor: Calcium/calmodulin-dependent protein kinase kinase 1, N-[2-OXO-3-((E)-PHENYL{[4-(PIPERIDIN-1-YLMETHYL)PHENYL]IMINO}METHYL)-2,6-DIHYDRO-1H-INDOL-5-YL]ETHANESULFONAMIDE, THIOCYANATE ION, ... (5 entities in total)
• Functional Keywords: protein kinase domain, structural genomics, structural genomics consortium, sgc, psi-biology, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 2
• Total formula weight: 66558.87

Authors

Santiago, A.S.,Counago, R.M.,dos Reis, C.V.,Ramos, P.Z.,Silva, P.N.B.,Drewry, D.,Elkins, J.M.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Structural Genomics Consortium (SGC) (deposition date: 2018-02-07, release date: 2018-03-07, Last modification date: 2023-10-04)

• Primary citation: Santiago, A.S.,Counago, R.M.,dos Reis, C.V.,Ramos, P.Z.,Drewry, D.,Elkins, J.M.,Massirer, K.B.,Arruda, P.,Edwards, A.M.; Crystal Structure of the Human CAMKK1A in complex with Hesperadin; To be Published,

Experimental method

X-RAY DIFFRACTION (2.1 Å)