6BRC
Crystal Structure of the Human CAMKK2B in complex with AP26113-analog (ALK-IN-1)
Summary for 6BRC
Entry DOI | 10.2210/pdb6brc/pdb |
Descriptor | Calcium/calmodulin-dependent protein kinase kinase 2, 5-chloro-N~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-N~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamine, SODIUM ION, ... (4 entities in total) |
Functional Keywords | transferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase inhibitor complex, transferase-transferase inhbitor complex, transferase/transferase inhbitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 67335.52 |
Authors | Counago, R.M.,dos Reis, C.V.,de Souza, G.P.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) (deposition date: 2017-11-30, release date: 2017-12-13, Last modification date: 2023-10-04) |
Primary citation | Counago, R.M.,dos Reis, C.V.,de Souza, G.P.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) Crystal Structure of the Human CAMKK2B in complex with AP26113-analog (ALK-IN-1) To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
Download full validation report