6BOZ
Structure of human SETD8 in complex with covalent inhibitor MS4138
Summary for 6BOZ
Entry DOI | 10.2210/pdb6boz/pdb |
Descriptor | N-lysine methyltransferase KMT5A, 1,2-ETHANEDIOL, N-(3-{[7-(2-aminoethoxy)-6-methoxy-2-(pyrrolidin-1-yl)quinazolin-4-yl]amino}propyl)prop-2-enamide, ... (4 entities in total) |
Functional Keywords | protein-small molecule inhibitor complex, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 44387.83 |
Authors | Babault, N.,Anqi, M.,Jin, J. (deposition date: 2017-11-21, release date: 2019-05-01, Last modification date: 2019-12-04) |
Primary citation | Chen, S.,Wiewiora, R.P.,Meng, F.,Babault, N.,Ma, A.,Yu, W.,Qian, K.,Hu, H.,Zou, H.,Wang, J.,Fan, S.,Blum, G.,Pittella-Silva, F.,Beauchamp, K.A.,Tempel, W.,Jiang, H.,Chen, K.,Skene, R.J.,Zheng, Y.G.,Brown, P.J.,Jin, J.,Luo, C.,Chodera, J.D.,Luo, M. The dynamic conformational landscape of the protein methyltransferase SETD8. Elife, 8:-, 2019 Cited by PubMed: 31081496DOI: 10.7554/eLife.45403 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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