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6BLE

Crystal Structure of the Human CAMKK2B in complex with CP673451

Summary for 6BLE
Entry DOI10.2210/pdb6ble/pdb
DescriptorCalcium/calmodulin-dependent protein kinase kinase 2, 1-{2-[5-(2-methoxyethoxy)-1H-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine, GLYCEROL, ... (4 entities in total)
Functional Keywordstransferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase inhibitor complex
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight33636.85
Authors
Counago, R.M.,dos Reis, C.V.,de Souza, G.P.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) (deposition date: 2017-11-10, release date: 2017-11-29, Last modification date: 2023-10-04)
Primary citationCounago, R.M.,dos Reis, C.V.,de Souza, G.P.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.
Crystal Structure of the Human CAMKK2B in complex with CP673451
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

236620

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