6AG3
Crystal structure of uPA in complex with 3,5-bis(azanyl)-N-carbamimidoyl-6-(2,4-dimethoxypyrimidin-5-yl)pyrazine-2-carboxamide
Summary for 6AG3
Entry DOI | 10.2210/pdb6ag3/pdb |
Descriptor | Urokinase-type plasminogen activator, 3,5-bis(azanyl)-N-carbamimidoyl-6-(2,4-dimethoxypyrimidin-5-yl)pyrazine-2-carboxamide (3 entities in total) |
Functional Keywords | urokinase, amiloride, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 28775.68 |
Authors | Buckley, B.,Jiang, L.G.,Majed, H.,Huang, M.D.,Kelso, M.,Ranson, M. (deposition date: 2018-08-09, release date: 2019-09-18, Last modification date: 2023-11-22) |
Primary citation | Buckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M. uPA-HMA To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.48 Å) |
Structure validation
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