6ZCY
SYK Kinase domain in complex with diamine inhibitor 16
Summary for 6ZCY
Entry DOI | 10.2210/pdb6zcy/pdb |
Descriptor | Tyrosine-protein kinase SYK, ~{N},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{R})-pyrrolidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide (3 entities in total) |
Functional Keywords | syk kinase transferase inhibitor, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 35327.48 |
Authors | Read, J.A. (deposition date: 2020-06-12, release date: 2021-06-23, Last modification date: 2024-01-24) |
Primary citation | Read, J.A. SYK Kinase domain in complex with azabenzimidazole inhibitor 16 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.81 Å) |
Structure validation
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