6Y3W
Ternary complex of 14-3-3 sigma (C38N), Estrogen Related Receptor gamma (DBD) phosphopeptide, and disulfide PPI stabilizer 1
Summary for 6Y3W
Entry DOI | 10.2210/pdb6y3w/pdb |
Descriptor | 14-3-3 protein sigma, Estrogen Related Receptor gamma phosphopetide, MAGNESIUM ION, ... (6 entities in total) |
Functional Keywords | 14-3-3, erry phosphopeptide, disulfide, stabilization, peptide binding protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 28090.89 |
Authors | Somsen, B.A.,Ottmann, C. (deposition date: 2020-02-19, release date: 2020-11-18, Last modification date: 2024-01-24) |
Primary citation | Sijbesma, E.,Somsen, B.A.,Miley, G.P.,Leijten-van de Gevel, I.A.,Brunsveld, L.,Arkin, M.R.,Ottmann, C. Fluorescence Anisotropy-Based Tethering for Discovery of Protein-Protein Interaction Stabilizers. Acs Chem.Biol., 15:3143-3148, 2020 Cited by PubMed: 33196173DOI: 10.1021/acschembio.0c00646 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.34 Å) |
Structure validation
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