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6P39

Crystal Structure Analysis of TAF1 Bromodomain

Summary for 6P39
Entry DOI10.2210/pdb6p39/pdb
DescriptorTranscription initiation factor TFIID subunit 1, 3-methoxy-4-{[(6aR)-5-methyl-6-oxo-6,6a,7,8,9,10-hexahydro-5H-dipyrido[1,2-a:3',2'-e]pyrazin-2-yl]amino}-N-(1-methylpiperidin-4-yl)benzamide (2 entities in total)
Functional Keywordskinase, bromodomain, inhibitor, transcription, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight16476.49
Authors
Seo, H.-S.,Dhe-Paganon, S. (deposition date: 2019-05-23, release date: 2020-05-27, Last modification date: 2023-10-11)
Primary citationSeo, H.-S.,Dhe-Paganon, S.
Crystal Structure Analysis of TAF1 Bromodomain
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.941 Å)
Structure validation

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