6N8G
IRAK4 bound to benzoxazole compound
Summary for 6N8G
Entry DOI | 10.2210/pdb6n8g/pdb |
Descriptor | Interleukin-1 receptor-associated kinase 4, N-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide (3 entities in total) |
Functional Keywords | protein kinase, irak4, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 136309.53 |
Authors | Larsen, N.A.,Bloudoff, K.,Subramanian, V.,Dobrzanska, M.,Gluza, K. (deposition date: 2018-11-29, release date: 2018-12-12) |
Primary citation | Larsen, N.A.,Gluza, K. To be published To Be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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