6KEE
Crystal structure of BRD4 Bromodomain1 with an inhibitor
Summary for 6KEE
Entry DOI | 10.2210/pdb6kee/pdb |
Descriptor | Bromodomain-containing protein 4, 6-[2-[2,4-bis(fluoranyl)phenoxy]-5-(methylsulfonylmethyl)pyridin-3-yl]-8-methyl-2H-pyrrolo[1,2-a]pyrazin-1-one (3 entities in total) |
Functional Keywords | antitumor, bet proteins, bromodomain inhibitor, epigenetic readers, antitumor protein, transcription |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15544.82 |
Authors | |
Primary citation | Xiao, S.,Li, Z.,Chen, S.,Zhou, B.,Luo, C. Crystal structure of BRD4 Bromodomain1 with an inhibitor To be published, |
Experimental method | X-RAY DIFFRACTION (2.12154661767 Å) |
Structure validation
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