6J3B
Crystal structure of human DHODH in complex with inhibitor 1289
Summary for 6J3B
Entry DOI | 10.2210/pdb6j3b/pdb |
Descriptor | Dihydroorotate dehydrogenase (quinone), mitochondrial, SODIUM ION, SULFATE ION, ... (11 entities in total) |
Functional Keywords | dhodh, inhibitor, complex, oxidoreductase, oxidoreductase-oxidoreductase inhibitor complex, oxidoreductase/oxidoreductase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 42221.84 |
Authors | |
Primary citation | Zeng, T.,Zuo, Z.,Luo, Y.,Zhao, Y.,Yu, Y.,Chen, Q. A novel series of human dihydroorotate dehydrogenase inhibitors discovered by in vitro screening: inhibition activity and crystallographic binding mode. Febs Open Bio, 9:1348-1354, 2019 Cited by PubMed: 31087527DOI: 10.1002/2211-5463.12658 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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