6F8B
LasB bound to thiol based inhibitor
Summary for 6F8B
Entry DOI | 10.2210/pdb6f8b/pdb |
Descriptor | Elastase, CALCIUM ION, ZINC ION, ... (5 entities in total) |
Functional Keywords | lasb, inhibitor, hydrolase |
Biological source | Pseudomonas aeruginosa |
Total number of polymer chains | 1 |
Total formula weight | 33753.25 |
Authors | Koehnke, J.,Sikandar, A. (deposition date: 2017-12-12, release date: 2018-03-28, Last modification date: 2024-01-17) |
Primary citation | Kany, A.M.,Sikandar, A.,Haupenthal, J.,Yahiaoui, S.,Maurer, C.K.,Proschak, E.,Kohnke, J.,Hartmann, R.W. Binding Mode Characterization and Early in Vivo Evaluation of Fragment-Like Thiols as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa. ACS Infect Dis, 4:988-997, 2018 Cited by PubMed: 29485268DOI: 10.1021/acsinfecdis.8b00010 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.3 Å) |
Structure validation
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