6ETJ
HUMAN PFKFB3 IN COMPLEX WITH KAN0438241
Summary for 6ETJ
Entry DOI | 10.2210/pdb6etj/pdb |
Descriptor | 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3, DIMETHYL SULFOXIDE, 6-O-phosphono-beta-D-fructofuranose, ... (6 entities in total) |
Functional Keywords | dna damage repair, homologous recombination, glycolysis, nucleotide metabolism, pfkfb3, antitumor protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 60941.96 |
Authors | Gustafsson, N.M.S.,Lundback, T.,Farnegardh, K.,Groth, P.,Wiitta, E.,Jonsson, M.,Hallberg, K.,Pennisi, R.,Huguet Ninou, A.,Martinsson, J.,Norstrom, C.,Schultz, J.,Andersson, M.,Markova, N.,Marttila, P.,Norin, M.,Olin, T.,Helleday, T. (deposition date: 2017-10-26, release date: 2018-11-07, Last modification date: 2020-07-29) |
Primary citation | Gustafsson, N.M.S.,Farnegardh, K.,Bonagas, N.,Ninou, A.H.,Groth, P.,Wiita, E.,Jonsson, M.,Hallberg, K.,Lehto, J.,Pennisi, R.,Martinsson, J.,Norstrom, C.,Hollers, J.,Schultz, J.,Andersson, M.,Markova, N.,Marttila, P.,Kim, B.,Norin, M.,Olin, T.,Helleday, T. Targeting PFKFB3 radiosensitizes cancer cells and suppresses homologous recombination. Nat Commun, 9:3872-3872, 2018 Cited by PubMed: 30250201DOI: 10.1038/s41467-018-06287-x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.51 Å) |
Structure validation
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