5Z14
Crystal structure of human TLR8 in complex with CU-CPT9a
Summary for 5Z14
Entry DOI | 10.2210/pdb5z14/pdb |
Related | 5WYX 5WYZ |
Descriptor | Toll-like receptor 8, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total) |
Functional Keywords | immune system |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 190708.50 |
Authors | Tanji, H.,Ohto, U.,Shimizu, T. (deposition date: 2017-12-25, release date: 2018-07-04, Last modification date: 2020-07-29) |
Primary citation | Hu, Z.,Zhang, S.,Tanji, H.,Jiang, S.,Li, J.,Sakaniwa, K.,Jin, J.,Bian, Y.,Ohto, U.,Shimizu, T.,Yin, H. Inhibition of Toll-like Receptor 8 by Specifically Targeting a Unique Allosteric Site and Locking Its Resting State To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
Download full validation report