5YOU
Crystal structure of BRD4-BD1 bound with hjp64
Summary for 5YOU
Entry DOI | 10.2210/pdb5you/pdb |
Descriptor | Bromodomain-containing protein 4, (3~{R})-4-cyclopropyl-~{N},1,3-trimethyl-~{N}-(4-methylphenyl)-2-oxidanylidene-3~{H}-quinoxaline-6-carboxamide (3 entities in total) |
Functional Keywords | bromodomain, transcription-inhibitor complex, transcription/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15462.83 |
Authors | Bing, X.,Jianping, H.,Yanlian, L.,Danyan, C. (deposition date: 2017-10-31, release date: 2018-11-07, Last modification date: 2024-03-27) |
Primary citation | Bing, X.,Jianping, H.,Yanlian, L.,Danyan, C. Crystal structure of BRD4-BD1 bound with hjp64 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.503 Å) |
Structure validation
Download full validation report