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5Y2I

Phosphoglycerate mutase 1 (PGAM1) complexed with its inhibitor PGMI-004A

Summary for 5Y2I
Entry DOI10.2210/pdb5y2i/pdb
DescriptorPhosphoglycerate mutase 1, 3,4-bis(oxidanyl)-9,10-bis(oxidanylidene)-~{N}-[4-(trifluoromethyl)phenyl]anthracene-2-sulfonamide, CHLORIDE ION, ... (5 entities in total)
Functional Keywordsphosphoglycerate mutase, isomerase-inhibitor complex, isomerase/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight60528.28
Authors
Jiang, L.,Zhou, L. (deposition date: 2017-07-26, release date: 2018-08-08, Last modification date: 2023-11-22)
Primary citationJiang, L.,Zhou, L.
Phosphoglycerate mutase 1 (PGAM1) complexed with its inhibitor PGMI-004A
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.917 Å)
Structure validation

217705

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