5XI4
BRD4 bound with compound Bdi4
Summary for 5XI4
Entry DOI | 10.2210/pdb5xi4/pdb |
Descriptor | Bromodomain-containing protein 4, (3~{S})-4-cyclopropyl-1,3-dimethyl-6-[[(1~{S})-1-(4-methylphenyl)ethyl]amino]-3~{H}-quinoxalin-2-one (3 entities in total) |
Functional Keywords | chromatin regulator, transcription-inhibitor complex, transcription/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: O60885 |
Total number of polymer chains | 1 |
Total formula weight | 15103.54 |
Authors | |
Primary citation | Xiong, B.,Cao, D.,Li, Y. BRD4 bound with compound Bdi4 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.486 Å) |
Structure validation
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