5XI2

BRD4 bound with compound Bdi2

Summary for 5XI2

• Entry DOI: 10.2210/pdb5xi2/pdb
• Descriptor: Bromodomain-containing protein 4, (3~{R})-4-cyclopropyl-1,3-dimethyl-6-[[(1~{S})-1-(4-methylphenyl)ethyl]amino]-3~{H}-quinoxalin-2-one (3 entities in total)
• Functional Keywords: chromatin regulator, transcription-inhibitor complex, transcription/inhibitor
• Biological source: Homo sapiens (Human)
• Cellular location: Nucleus: O60885
• Total number of polymer chains: 1
• Total formula weight: 15103.54

Authors

Xiong, B.,Cao, D.,Li, Y. (deposition date: 2017-04-25, release date: 2018-05-02, Last modification date: 2024-03-27)

• Primary citation: Xiong, B.,Cao, D.,Li, Y.; BRD4 bound with compound Bdi2; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.909 Å)