5UNG
XFEL structure of human angiotensin II type 2 receptor (Orthorhombic form) in complex with compound 1 (N-benzyl-N-(2-ethyl-4-oxo-3-{[2'-(2H-tetrazol-5-yl)[1,1'-biphenyl]-4-yl] methyl}-3,4-dihydroquinazolin-6-yl)thiophene-2-carboxamide)
5UNG の概要
エントリーDOI | 10.2210/pdb5ung/pdb |
関連するPDBエントリー | 5UNF 5UNH |
分子名称 | Chimera protein of Type-2 angiotensin II receptor and Soluble cytochrome b562, N-benzyl-N-(2-ethyl-4-oxo-3-{[2'-(2H-tetrazol-5-yl)[1,1'-biphenyl]-4-yl]methyl}-3,4-dihydroquinazolin-6-yl)thiophene-2-carboxamide, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, ... (5 entities in total) |
機能のキーワード | human angiotensin ii receptor complex, gpcr signaling, gpcr, bril, membrane protein, lcp, xfel, blood pressure regulation, orthorhombic crystal, compound 1 (cpd 1), signaling protein |
由来する生物種 | Escherichia coli 詳細 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 47769.26 |
構造登録者 | Zhang, H.,Han, G.W.,Batyuk, A.,Ishchenko, A.,White, K.L.,Patel, N.,Sadybekov, A.,Zamlynny, B.,Rudd, M.T.,Hollenstein, K.,Tolstikova, A.,White, T.A.,Hunter, M.S.,Weierstall, U.,Liu, W.,Babaoglu, K.,Moore, E.L.,Katz, R.D.,Shipman, J.M.,Garcia-Calvo, M.,Sharma, S.,Sheth, P.,Soisson, S.M.,Stevens, R.C.,Katritch, V.,Cherezov, V. (登録日: 2017-01-30, 公開日: 2017-04-05, 最終更新日: 2023-10-04) |
主引用文献 | Zhang, H.,Han, G.W.,Batyuk, A.,Ishchenko, A.,White, K.L.,Patel, N.,Sadybekov, A.,Zamlynny, B.,Rudd, M.T.,Hollenstein, K.,Tolstikova, A.,White, T.A.,Hunter, M.S.,Weierstall, U.,Liu, W.,Babaoglu, K.,Moore, E.L.,Katz, R.D.,Shipman, J.M.,Garcia-Calvo, M.,Sharma, S.,Sheth, P.,Soisson, S.M.,Stevens, R.C.,Katritch, V.,Cherezov, V. Structural basis for selectivity and diversity in angiotensin II receptors. Nature, 544:327-332, 2017 Cited by PubMed: 28379944DOI: 10.1038/nature22035 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.8 Å) |
構造検証レポート
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