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5UEQ

BRD4_BD2_A-1390146

Summary for 5UEQ
Entry DOI10.2210/pdb5ueq/pdb
Related5UEO 5UEP 5UER 5UES 5UET 5UEU 5UEV 5UEW 5UEX 5UEY 5UEZ 5UF0
DescriptorBromodomain-containing protein 4, N-[3-(7-methyl-1-oxo-2,6-dihydro-1H-pyrrolo[3,4-d]pyridazin-5-yl)-4-phenoxyphenyl]ethanesulfonamide (3 entities in total)
Functional Keywordssignaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains1
Total formula weight13231.41
Authors
Park, C.H. (deposition date: 2017-01-03, release date: 2017-06-14, Last modification date: 2024-04-03)
Primary citationPark, C.H.
Complex structure of BRD4_BD2_A-1390146
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

218500

PDB entries from 2024-04-17

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