5TUI
Crystal structure of tetracycline destructase Tet(50) in complex with chlortetracycline
Summary for 5TUI
Entry DOI | 10.2210/pdb5tui/pdb |
Related | 5TUE 5TUF 5TUK 5TUL 5TUM |
Descriptor | Tetracycline destructase Tet(50), SULFATE ION, FLAVIN-ADENINE DINUCLEOTIDE, ... (5 entities in total) |
Functional Keywords | fad-binding, tetracycline-inactivating, oxidoreductase activity, oxidoreductase |
Biological source | uncultured bacterium |
Total number of polymer chains | 2 |
Total formula weight | 94590.80 |
Authors | Park, J.,Tolia, N.H. (deposition date: 2016-11-06, release date: 2017-05-10, Last modification date: 2024-03-06) |
Primary citation | Park, J.,Gasparrini, A.J.,Reck, M.R.,Symister, C.T.,Elliott, J.L.,Vogel, J.P.,Wencewicz, T.A.,Dantas, G.,Tolia, N.H. Plasticity, dynamics, and inhibition of emerging tetracycline resistance enzymes. Nat. Chem. Biol., 13:730-736, 2017 Cited by PubMed: 28481346DOI: 10.1038/nchembio.2376 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
Download full validation report