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5TS8

Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 5,6-DIBROMOBENZOTRIAZOLE

Summary for 5TS8
Entry DOI10.2210/pdb5ts8/pdb
Related1DAW 1J91 1P5E 2OXY 4KWP 4RKL
DescriptorProtein kinase CK2 catalytic subunit CK2 alpha-3, 5,6-DIBROMOBENZOTRIAZOLE, L(+)-TARTARIC ACID, ... (10 entities in total)
Functional Keywordsck2, casein kinase 2, inhibitor, bromo-benzotriazole, transferase-transferase inhibitor complex, halogen bond, transferase/transferase inhibitor
Biological sourceZea mays
Total number of polymer chains1
Total formula weight41490.89
Authors
Winiewska, M.,Kucinska, K.,Czapinska, H.,Piasecka, A.,Bochtler, M.,Poznanski, J. (deposition date: 2016-10-28, release date: 2018-01-17, Last modification date: 2024-01-17)
Primary citationWiniewska, M.,Kucinska, K.,Czapinska, H.,Piasecka, A.,Bochtler, M.,Poznanski, J.
STRUCTURAL AND THERMODYNAMIC ANALYSIS OF 5,6-DIBROMOBENZOTRIAZOLE BINDING TO CASEIN KINASE 2 ALPHA
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.45 Å)
Structure validation

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