5TEH
c-Src V281C kinase domain in complex with Rao-IV-156
Summary for 5TEH
Entry DOI | 10.2210/pdb5teh/pdb |
Related | 5SWH |
Descriptor | Proto-oncogene tyrosine-protein kinase Src, (2S)-3-[4-amino-7-(2-methoxyethyl)-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyano-N-(propan-2-yl)propanamide (3 entities in total) |
Functional Keywords | ac helix out, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Gallus gallus (Chicken) |
Total number of polymer chains | 2 |
Total formula weight | 66458.46 |
Authors | Dieter, E.M.,Merritt, E.A.,Maly, D.J. (deposition date: 2016-09-21, release date: 2017-09-27, Last modification date: 2023-10-04) |
Primary citation | Register, A.C.,Maly, D.J. A combined approach reveals a regulatory mechanism coupling Src's kinase activity, localization, and phosphotransferase-independent functions Mol.Cell, 2019:-, |
Experimental method | X-RAY DIFFRACTION (2.99 Å) |
Structure validation
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