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5S5K

Tubulin-Z2472938267-complex

Summary for 5S5K
Entry DOI10.2210/pdb5s5k/pdb
Group depositionXChem fragment screening on T2R-TTL (G_1002173)
DescriptorTubulin alpha-1B chain, 1-[2-(2-oxidanylidenepyrrolidin-1-yl)ethyl]-3-phenyl-urea, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... (12 entities in total)
Functional Keywordscell cycle, tubulin fold, cytoskeleton, microtubule
Biological sourceRattus norvegicus (Rat)
More
Total number of polymer chains6
Total formula weight264793.66
Authors
Muehlethaler, T.,Gioia, D.,Prota, A.E.,Sharpe, M.E.,Cavalli, A.,Steinmetz, M.O. (deposition date: 2020-11-08, release date: 2021-06-30, Last modification date: 2024-03-06)
Primary citationMuhlethaler, T.,Gioia, D.,Prota, A.E.,Sharpe, M.E.,Cavalli, A.,Steinmetz, M.O.
Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60:13331-13342, 2021
Cited by
PubMed: 33951246
DOI: 10.1002/anie.202100273
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.41 Å)
Structure validation

217705

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