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5LV4

Crystal structure of mouse PRMT6 in complex with inhibitor LH1236

Summary for 5LV4
Entry DOI10.2210/pdb5lv4/pdb
DescriptorProtein arginine N-methyltransferase 6, (2~{R})-4-[[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl-[[4-azanyl-1-(methoxymethyl)-2-oxidanylidene-pyrimidin-5-yl]methyl]amino]-2-azanyl-butanoic acid (3 entities in total)
Functional Keywordstransferase, s-adenosyl-l-methionine
Biological sourceMus musculus (House Mouse)
Cellular locationNucleus : Q6NZB1
Total number of polymer chains1
Total formula weight45131.67
Authors
Cura, V.,Marechal, N.,Troffer-Charlier, N.,Halby, L.,Arimondo, P.,Bonnefond, L.,Cavarelli, J. (deposition date: 2016-09-12, release date: 2017-09-20, Last modification date: 2024-01-17)
Primary citationHalby, L.,Marechal, N.,Pechalrieu, D.,Cura, V.,Franchini, D.M.,Faux, C.,Alby, F.,Troffer-Charlier, N.,Kudithipudi, S.,Jeltsch, A.,Aouadi, W.,Decroly, E.,Guillemot, J.C.,Page, P.,Ferroud, C.,Bonnefond, L.,Guianvarc'h, D.,Cavarelli, J.,Arimondo, P.B.
Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors.
Philos. Trans. R. Soc. Lond., B, Biol. Sci., 373:-, 2018
Cited by
PubMed: 29685976
DOI: 10.1098/rstb.2017.0072
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.66 Å)
Structure validation

217705

數據於2024-03-27公開中

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