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5K20

Caspase-7 S239E Phosphomimetic

Summary for 5K20
Entry DOI10.2210/pdb5k20/pdb
Related1K86 3IBF 3R5K 3S8E
DescriptorCaspase-7 large subunit, Caspase-7 small subunit, FORMIC ACID, ... (4 entities in total)
Functional Keywordsprotease, phosphomimetic, pak2, phosphorylation, hydrolase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains4
Total formula weight71048.15
Authors
Eron, S.J.,Hardy, J.A. (deposition date: 2016-05-18, release date: 2017-01-11, Last modification date: 2023-09-27)
Primary citationEron, S.J.,Hardy, J.A.
PAK2 Phosphorylation Inhibits Caspase-7 by Two Divergent Mechanisms: Slowing Activation and Blocking Substrate Binding
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

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