5J7W
Enterococcus faecalis thymidylate synthase complex with methotrexate
Summary for 5J7W
Entry DOI | 10.2210/pdb5j7w/pdb |
Descriptor | Thymidylate synthase, SULFATE ION, METHOTREXATE, ... (4 entities in total) |
Functional Keywords | enterococcus faecalis, thymidylate synthase, methotrexate, complex, transferase |
Biological source | Enterococcus faecalis |
Cellular location | Cytoplasm : Q834R3 |
Total number of polymer chains | 4 |
Total formula weight | 146837.04 |
Authors | Mangani, S.,Pozzi, C. (deposition date: 2016-04-07, release date: 2016-09-28, Last modification date: 2024-05-08) |
Primary citation | Catalano, A.,Luciani, R.,Carocci, A.,Cortesi, D.,Pozzi, C.,Borsari, C.,Ferrari, S.,Mangani, S. X-ray crystal structures of Enterococcus faecalis thymidylate synthase with folate binding site inhibitors. Eur.J.Med.Chem., 123:649-664, 2016 Cited by PubMed: 27517810DOI: 10.1016/j.ejmech.2016.07.066 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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