5FX5
Novel inhibitors of human rhinovirus 3C protease
5FX5 の概要
エントリーDOI | 10.2210/pdb5fx5/pdb |
関連するPDBエントリー | 5FX6 |
分子名称 | RHINOVIRUS 3C PROTEASE, GLYCEROL, TETRAETHYLENE GLYCOL, ... (6 entities in total) |
機能のキーワード | transferase |
由来する生物種 | HUMAN RHINOVIRUS 2 (HRV2) |
細胞内の位置 | Capsid protein VP0: Virion . Capsid protein VP4: Virion . Capsid protein VP2: Virion . Capsid protein VP3: Virion . Capsid protein VP1: Virion . Protein 2B: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 2C: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 3A: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 3AB: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Viral protein genome-linked: Virion . Protease 3C: Host cytoplasm . Protein 3CD: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . RNA-directed RNA polymerase: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side : P04936 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 21264.09 |
構造登録者 | Kawatkar, S.,Ek, M.,Hoesch, V.,Gagnon, M.,Nilsson, E.,Lister, T.,Olsson, L.,Patel, J.,Yu, Q. (登録日: 2016-02-24, 公開日: 2016-06-22, 最終更新日: 2024-01-10) |
主引用文献 | Kawatkar, S.P.,Gagnon, M.,Hoesch, V.,Tiong-Yip, C.,Johnson, K.,Ek, M.,Nilsson, E.,Lister, T.,Olsson, L.,Patel, J.,Yu, Q. Design and Structure-Activity Relationships of Novel Inhibitors of Human Rhinovirus 3C Protease. Bioorg.Med.Chem.Lett., 26:3248-, 2016 Cited by PubMed: 27265257DOI: 10.1016/J.BMCL.2016.05.066 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.7 Å) |
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