5F1R
The Transcriptional Regulator PrfA from Listeria Monocytogenes in complex with a ring-fused 2-pyridone (C10)
Summary for 5F1R
Entry DOI | 10.2210/pdb5f1r/pdb |
Related | 2BEO |
Descriptor | Listeriolysin regulatory protein, (3~{R})-8-cyclopropyl-7-(naphthalen-1-ylmethyl)-5-oxidanylidene-2,3-dihydro-[1,3]thiazolo[3,2-a]pyridine-3-carboxylic acid (3 entities in total) |
Functional Keywords | dna binding protein, prfa, 2-pyridones, virulence |
Biological source | Listeria monocytogenes serovar 1/2a (strain ATCC BAA-679 / EGD-e) |
Total number of polymer chains | 2 |
Total formula weight | 55413.69 |
Authors | Begum, A.,Grundstrom, C.,Good, J.A.D.,Andersson, C.,ALmqvist, F.,Johansson, J.,Sauer, U.H.,Sauer-Eriksson, A.E. (deposition date: 2015-11-30, release date: 2016-03-16, Last modification date: 2024-01-10) |
Primary citation | Good, J.A.,Andersson, C.,Hansen, S.,Wall, J.,Krishnan, K.S.,Begum, A.,Grundstrom, C.,Niemiec, M.S.,Vaitkevicius, K.,Chorell, E.,Wittung-Stafshede, P.,Sauer, U.H.,Sauer-Eriksson, A.E.,Almqvist, F.,Johansson, J. Attenuating Listeria monocytogenes Virulence by Targeting the Regulatory Protein PrfA. Cell Chem Biol, 23:404-414, 2016 Cited by PubMed: 26991105DOI: 10.1016/j.chembiol.2016.02.013 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.25 Å) |
Structure validation
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