5EQI
Human GLUT1 in complex with Cytochalasin B
Summary for 5EQI
Entry DOI | 10.2210/pdb5eqi/pdb |
Related | 5EQG 5EQH |
Descriptor | Solute carrier family 2, facilitated glucose transporter member 1, Cytochalasin B (2 entities in total) |
Functional Keywords | mfs transporter, glucose transporter, transport protein-inhibitor complex, transport protein/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 54605.00 |
Authors | Kapoor, K.,Finer-Moore, J.,Pedersen, B.P.,Caboni, L.,Waight, A.B.,Hillig, R.,Bringmann, P.,Heisler, I.,Muller, T.,Siebeneicher, H.,Stroud, R.M. (deposition date: 2015-11-12, release date: 2016-04-13, Last modification date: 2023-09-27) |
Primary citation | Kapoor, K.,Finer-Moore, J.S.,Pedersen, B.P.,Caboni, L.,Waight, A.,Hillig, R.C.,Bringmann, P.,Heisler, I.,Muller, T.,Siebeneicher, H.,Stroud, R.M. Mechanism of inhibition of human glucose transporter GLUT1 is conserved between cytochalasin B and phenylalanine amides. Proc.Natl.Acad.Sci.USA, 113:4711-4716, 2016 Cited by PubMed: 27078104DOI: 10.1073/pnas.1603735113 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.002 Å) |
Structure validation
Download full validation report