5E95
Crystal Structure of Mb(NS1)/H-Ras Complex
Summary for 5E95
Entry DOI | 10.2210/pdb5e95/pdb |
Descriptor | Mb(NS1), GTPase HRas, GUANOSINE-5'-DIPHOSPHATE, ... (5 entities in total) |
Functional Keywords | h-ras, monobody, inhibitor, complex, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Homo sapiens More |
Total number of polymer chains | 2 |
Total formula weight | 29907.47 |
Authors | Eguchi, R.R.,Sha, F.,Gupta, A.,Koide, A.,Koide, S. (deposition date: 2015-10-14, release date: 2016-11-02, Last modification date: 2023-09-27) |
Primary citation | Spencer-Smith, R.,Koide, A.,Zhou, Y.,Eguchi, R.R.,Sha, F.,Gajwani, P.,Santana, D.,Gupta, A.,Jacobs, M.,Herrero-Garcia, E.,Cobbert, J.,Lavoie, H.,Smith, M.,Rajakulendran, T.,Dowdell, E.,Okur, M.N.,Dementieva, I.,Sicheri, F.,Therrien, M.,Hancock, J.F.,Ikura, M.,Koide, S.,O'Bryan, J.P. Inhibition of RAS function through targeting an allosteric regulatory site. Nat. Chem. Biol., 13:62-68, 2017 Cited by PubMed: 27820802DOI: 10.1038/nchembio.2231 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.402 Å) |
Structure validation
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