5E16
Co-crystal structure of the N-termial cGMP binding domain of Plasmodium falciparum PKG with cGMP
Summary for 5E16
Entry DOI | 10.2210/pdb5e16/pdb |
Descriptor | CGMP-dependent protein kinase, CYCLIC GUANOSINE MONOPHOSPHATE (3 entities in total) |
Functional Keywords | kinase, cgmp binding domain, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Plasmodium falciparum |
Total number of polymer chains | 1 |
Total formula weight | 16423.28 |
Authors | El Bakkouri, M.,Walker, J.R.,Loppnau, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Hui, R.,Structural Genomics Consortium (SGC) (deposition date: 2015-09-29, release date: 2015-11-04, Last modification date: 2023-09-27) |
Primary citation | El Bakkouri, M.,Kouidmi, I.,Wernimont, A.K.,Amani, M.,Hutchinson, A.,Loppnau, P.,Kim, J.J.,Flueck, C.,Walker, J.R.,Seitova, A.,Senisterra, G.,Kakihara, Y.,Kim, C.,Blackman, M.J.,Calmettes, C.,Baker, D.A.,Hui, R. Structures of the cGMP-dependent protein kinase in malaria parasites reveal a unique structural relay mechanism for activation. Proc.Natl.Acad.Sci.USA, 116:14164-14173, 2019 Cited by PubMed: 31239348DOI: 10.1073/pnas.1905558116 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.65 Å) |
Structure validation
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