5DQF
Horse Serum Albumin (ESA) in complex with Cetirizine
Summary for 5DQF
Entry DOI | 10.2210/pdb5dqf/pdb |
Descriptor | Serum albumin, TETRAETHYLENE GLYCOL, SULFATE ION, ... (7 entities in total) |
Functional Keywords | albumin, cetirizine, esa, nysgrc, structural genomics, psi-biology, new york structural genomics research consortium, transport protein |
Biological source | Equus caballus (Horse) |
Total number of polymer chains | 1 |
Total formula weight | 68077.17 |
Authors | Handing, K.B.,Shabalin, I.G.,Majorek, K.A.,Chruszcz, M.,Almo, S.C.,Minor, W.,New York Structural Genomics Research Consortium (NYSGRC) (deposition date: 2015-09-14, release date: 2015-12-23, Last modification date: 2023-09-27) |
Primary citation | Handing, K.B.,Shabalin, I.G.,Szlachta, K.,Majorek, K.A.,Minor, W. Crystal structure of equine serum albumin in complex with cetirizine reveals a novel drug binding site. Mol.Immunol., 71:143-151, 2016 Cited by PubMed: 26896718DOI: 10.1016/j.molimm.2016.02.003 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.15 Å) |
Structure validation
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