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5DM1

Crystal structure of the plantazolicin methyltransferase BpumL in complex with monoazolic desmethylPZN analog and SAH

Summary for 5DM1
Entry DOI10.2210/pdb5dm1/pdb
Related5DLY 5DM2 5DM4
DescriptorMethyltransferase domain family, prop-2-en-1-yl 2-[(1S)-1-amino-4-carbamimidamidobutyl]-1,3-thiazole-4-carboxylate, S-ADENOSYL-L-HOMOCYSTEINE, ... (5 entities in total)
Functional Keywordsn-methyltransferase, plantazolicin, monoazolic desmethylpzn analog, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceBacillus pumilus ATCC 7061
Total number of polymer chains1
Total formula weight31347.71
Authors
Hao, Y.,Nair, S.K. (deposition date: 2015-09-07, release date: 2015-09-23, Last modification date: 2024-03-06)
Primary citationHao, Y.,Blair, P.M.,Sharma, A.,Mitchell, D.A.,Nair, S.K.
Insights into methyltransferase specificity and bioactivity of derivatives of the antibiotic plantazolicin.
Acs Chem.Biol., 10:1209-1216, 2015
Cited by
PubMed: 25635336
DOI: 10.1021/cb501042a
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

217705

數據於2024-03-27公開中

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